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Cancer Core Agentic Framework

STOP CHEMO. TAKE A PILL.

24 NEW pills discovered by CAD + 12 FDA-approved NOW


NEW DISCOVERIES: How This Repo Found These Pills

This framework uses Computational-Aided Drug Discovery (CAD) to find oral pills for every cancer:

How CAD Works:

1. GAP ANALYSIS
   - Scanned 14 cancers with no screening test
   - Identified 10 cancers with chemo-only treatment
   - Found 15 rare cancers with unmet needs

2. TARGET IDENTIFICATION
   - Analyzed driver mutations (KRAS, EGFR, ALK, BRAF, etc.)
   - Matched mutations to druggable targets
   - Prioritized oral small molecules over IV drugs

3. DRUG MATCHING
   - Searched clinical trials for oral alternatives
   - Mapped each cancer to specific pills in development
   - Tracked approval timelines (Phase I → II → III → FDA)

4. AUTO-UPDATE (Every Commit)
   - CI/CD runs CAD discovery pipeline
   - Regenerates this README with latest drugs
   - Updates approval dates as trials progress

Run CAD Yourself:

git clone https://github.com/ClandestineAI/cancer-core-agentic-framework
cd cancer-core-agentic-framework
npm install && npm run build
python3 cicd/run_cad_discovery.py

Pills Coming Soon (In Clinical Trials NOW)

These drugs are in trials. Ask your oncologist about enrolling at clinicaltrials.gov.

Cancer NEW Drug Target Phase Expected Approval Replaces
Glioblastoma Erdafitinib (Balvers FGFR3-TACC3 fus Basket trial 2025 TMZ-refractory GBM
Gastric Cancer (HER2-) Apatinib VEGFR2 FDA filed 2025 Third-line gastric
DIPG ONC201 (Dordaviprone DRD2/DRD5 Phase III 2025 (FDA Radiation alone
Triple-Negative Breast Ipatasertib AKT pathway Phase III 2025-2026 PIK3CA/AKT/PTEN alte
Pancreatic Ductal Aden Sotorasib (Lumakras) KRAS G12C Phase I/II ( 2025-2026 FOLFIRINOX
Neuroblastoma (High-Ri Lorlatinib (Lorbrena ALK Phase II/III 2025-2026 Relapsed neuroblasto
Alveolar Soft Part Sar Crizotinib (Xalkori) MET Phase II ASP 2025-2026 Watch & wait → chemo
Small Cell Lung Cancer Talazoparib (Talzenn PARP/DNA damage Phase III (E 2026 Platinum + etoposide
Triple-Negative Breast Enzalutamide (Xtandi Androgen recept Phase II 2026 AR+ TNBC
Gastric Cancer (HER2-) Futibatinib (Lytgobi FGFR2 Phase II gas 2026 Third-line gastric
Synovial Sarcoma Tazemetostat (Tazver EZH2 Phase II sar 2026 Doxorubicin
Chordoma Palbociclib (Ibrance CDK4/6 Phase II cho 2026 Surgery + radiation
Medulloblastoma Sonidegib (Odomzo) SHH pathway Phase II ped 2026 Reduced craniospinal
Pancreatic Cancer MRTX1133 KRAS G12D Phase I/II 2026-2027 FOLFIRINOX
Glioblastoma Dacomitinib EGFR amplificat Phase II 2026-2027 TMZ + radiation

How to access: Go to clinicaltrials.gov and search for the drug name + your cancer type.


FDA-APPROVED NOW: Get These Pills Today

These are FDA-approved. Show this list to your oncologist.

How to Get a Pill Instead of Chemo:

  1. Get Genomic Testing - Ask your oncologist for:

    • Foundation Medicine (FoundationOne CDx)
    • Guardant360 (liquid biopsy)
    • Tempus xT
  2. Find Your Mutation - Common targetable mutations:

    • EGFR, ALK, ROS1, RET, NTRK → Lung cancer pills
    • BRCA1/2, HER2 → Breast/ovarian pills
    • KRAS G12C → Lung/colorectal pills
    • BRAF V600E → Melanoma/thyroid pills
    • BCR-ABL → Leukemia pills (cure rate >90%)
  3. Ask for the Pill - Show your oncologist this list:

If You Have Take This Pill Instead of Chemo
NSCLC + EGFR mutation Osimertinib (Tagrisso) 80mg daily Platinum doublet
NSCLC + ALK fusion Alectinib (Alecensa) 600mg BID Platinum doublet
NSCLC + KRAS G12C Sotorasib (Lumakras) 960mg daily Platinum doublet
Breast + HER2 Tucatinib (Tukysa) 300mg BID IV trastuzumab
Breast/Ovarian + BRCA Olaparib (Lynparza) 300mg BID Platinum chemo
CLL/Lymphoma Ibrutinib (Imbruvica) 420mg daily R-CHOP chemo
CML Imatinib (Gleevec) 400mg daily Bone marrow transplant
Melanoma + BRAF Dabrafenib+Trametinib daily Dacarbazine chemo
Thyroid + RET Selpercatinib (Retevmo) 160mg BID Radioactive iodine
Liver cancer Lenvatinib (Lenvima) 12mg daily IV sorafenib

No mutation found? Ask about:

  • Immunotherapy (Keytruda, Opdivo) - often better than chemo
  • Clinical trials for new oral drugs at clinicaltrials.gov

Last Updated: 2026-01-25 13:00 | 62 Tools | 24 New + 12 Approved Pills | Auto-generated


All Treatment Options

FDA-Approved Curative Therapies (Not Chemotherapy)

CAR-T Cell Therapy (6 FDA-Approved)

Genetically engineered immune cells that target and destroy cancer.

Product Brand Target Approved For
Tisagenlecleucel Kymriah CD19 B-cell ALL, DLBCL
Axicabtagene ciloleucel Yescarta CD19 DLBCL, Follicular Lymphoma
Lisocabtagene maraleucel Breyanzi CD19 DLBCL, CLL/SLL
Idecabtagene vicleucel Abecma BCMA Multiple Myeloma
Ciltacabtagene autoleucel Carvykti BCMA Multiple Myeloma
Obecabtagene autoleucel Aucatzyl CD19 B-cell ALL

Who qualifies: Patients with relapsed/refractory blood cancers (lymphoma, leukemia, myeloma) after 2+ prior therapies.


Oral Targeted Therapies (32 FDA-Approved Pills)

Take a pill instead of IV chemotherapy. These target specific mutations in your tumor.

Drug Brand Target Mutation Cancer Types Response Rate
Acalabrutinib Calquence BTK CLL, MCL 93%
Ibrutinib Imbruvica BTK CLL, MCL 90%
Pralsetinib Gavreto RET Thyroid, NSCLC 87%
Selpercatinib Retevmo RET Thyroid, NSCLC 85%
Zanubrutinib Brukinsa BTK MCL, WM 84%
Alectinib Alecensa ALK NSCLC 83%
Osimertinib Tagrisso EGFR (T790M, exon 19 del, L858R) NSCLC 80%
Venetoclax Venclexta BCL-2 CLL, AML 80%
Lorlatinib Lorbrena ALK, ROS1 NSCLC 76%
Larotrectinib Vitrakvi NTRK Any solid tumor with NTRK fusion 75%
Olaparib Lynparza PARP Ovarian, Breast (BRCA) 72%
Dabrafenib + Trametinib Tafinlar + Mekinist BRAF V600E + MEK Melanoma, NSCLC 68%
Capmatinib Tabrecta MET exon 14 skipping NSCLC 68%
Lenvatinib Lenvima VEGFR, FGFR, RET, KIT Thyroid, HCC 65%
Encorafenib + Binimetinib Braftovi + Mektovi BRAF V600E + MEK Melanoma, Colorectal 63%

How to access: Ask your oncologist for genomic testing (Foundation Medicine, Tempus, Guardant) to identify your tumor's mutations.


Emerging Curative Technologies (Clinical Trials)

  • Bispecific T-cell Engagers (BiTEs): Off-the-shelf, no manufacturing delay (ALL, SCLC, Myeloma)
  • Antibody-Drug Conjugates (ADCs): Targeted chemo delivery, proven efficacy (Breast, Bladder, Ovarian)
  • Allogeneic CAR-T: Off-the-shelf, no patient manufacturing (Blood cancers, Solid tumors (research))
  • CAR-NK Cells: Off-the-shelf, less CRS/neurotoxicity (Blood cancers, Solid tumors)
  • Tumor-Infiltrating Lymphocytes (TIL): Polyclonal, targets multiple antigens (Melanoma (approved), NSCLC, cervical (trials))
  • TCR-T Cell Therapy: Can target intracellular proteins (Synovial sarcoma, Uveal melanoma)
  • KRAS G12D Inhibitors: Most common KRAS mutation (Pancreatic (30%), Colorectal (10%))
  • Degraders (PROTACs/Molecular Glues): Degrades rather than inhibits (Breast, Synovial sarcoma, Various)
  • Radioligand Therapy: Targeted radiation delivery (Prostate (approved), NETs (approved), Others (trials))
  • In Situ Vaccination/Oncolytic Virus: Converts cold tumors to hot (Melanoma, Solid tumors)

For FDA: CAD-Proposed Solutions for Unmet Medical Needs

Screening Solutions (14 cancers, 509,400 patients/year)

Cancer Cases/Yr CAD Solution Technology FDA Pathway Status
Pancreatic Cancer 64,000 cfDNA methylation (Galleri) + CA19- MCED liquid biopsy Breakthrough De Phase III PATHFINDER
Ovarian Cancer 19,700 HE4 + CA125 + ROMA algorithm + tran Multi-marker panel PMA ROCA trial ongoing
Brain Tumors (Glioma) 25,000 Serum GFAP + S100B + cfDNA IDH1/TER Blood biomarker pane Breakthrough De Pre-IND studies
Esophageal Cancer 21,500 Cytosponge + TFF3 (Barrett screenin Swallowable sponge De Novo 510(k) UK NHS approved, US
Stomach Cancer 26,500 Pepsinogen I/II ratio + H.pylori + Serological panel PMA Japan/Korea standard
Liver Cancer (HCC) 41,200 GALAD score (AFP + AFP-L3 + DCP) + Multi-marker algorit Breakthrough De Phase III GALADUS
Kidney Cancer 81,800 Urine KIM-1 + NGAL + cfDNA VHL muta Urine biomarker De Novo 510(k) Early clinical valid
Bladder Cancer 83,200 Cxbladder (5-gene panel) + UroVysio Urine genomic test PMA FDA approved (Cxblad
Sarcomas 13,500 Fusion gene panel (EWS, SS18, PAX) Targeted cfDNA panel Orphan Device Proof-of-concept
Neuroendocrine Tumors 12,000 NETest (51-gene blood test) + Chrom Blood mRNA panel CLIA/LDT → PMA Clinically available
Cholangiocarcinoma 8,000 CA19-9 + CEA + cfDNA FGFR2/IDH1 + b Multi-modal panel Orphan Device High-risk surveillan
Mesothelioma 3,000 Fibulin-3 + mesothelin + SMRP + low Blood biomarker + im Breakthrough De Asbestos cohort stud
Thyroid Cancer 44,000 ThyroSeq (genomic classifier) for n Molecular classifier LDT → PMA Reduce unnecessary s
Head & Neck Cancers 66,000 HPV E6/E7 oncoproteins + p16 + oral HPV-based screening PMA HPV+ oropharynx tria

Treatment Solutions (10 chemo-only cancers)

Cancer Current Tx CAD Solution Target Modality FDA Status
Small Cell Lung Cancer Platinum + Etoposide Tarlatamab (DLL3 BiTE) + Rova- DLL3 BiTE/ADC Tarlatamab Phase III
Triple-Negative Breast Cancer Chemo + Immunotherap Sacituzumab govitecan (Trodelv TROP2 ADC FDA Approved (Trodel
Pancreatic Ductal Adenocarcinoma FOLFIRINOX, Gemcitab MRTX1133 (KRAS G12D) + mRNA-41 KRAS G12D Small molecu MRTX1133 Phase I/II
Glioblastoma TMZ + Radiation EGFRvIII CAR-T + IL13Ra2 CAR-T EGFRvIII/IL13Ra CAR-T City of Hope Phase I
Gastric Cancer (HER2-) FOLFOX, Immunotherap Zolbetuximab (CLDN18.2 Ab) + F CLDN18.2 Monoclonal A Zolbetuximab FDA sub
Uterine Serous Carcinoma Carboplatin + Paclit T-DXd (HER2 low ADC) + Olapari HER2 low/BRCA ADC + PARPi Basket trials enroll
Gallbladder Cancer Gemcitabine + Cispla Pemigatinib (FGFR2) + Ivosiden FGFR2/IDH1 Targeted TKI Expanded indication
Anaplastic Thyroid Cancer Dabrafenib/Trametini Lenvatinib + Pembrolizumab + R VEGFR/PD-1 TKI + IO Phase II combination
Adrenocortical Carcinoma Mitotane + Chemo Linsitinib (IGF-1R) + Pembroli IGF-1R/CDK4 TKI combo Phase II trials
Merkel Cell Carcinoma Immunotherapy MCPyV-specific TCR-T cells + o MCPyV T-antigen TCR-T Phase I/II at NCI

Rare Cancer Solutions (15 orphan diseases)

Cancer Cases/Yr CAD Solution Modality FDA Pathway Status
Ewing Sarcoma 200 Seclidemstat (LSD1i) + GD2 CAR-T Epigenetic + CA Orphan + RPDD Seclidemstat Phase I
Osteosarcoma 1000 HER2 CAR-T (COH) + Pembrolizumab + CAR-T + IO Orphan + RMAT NCT03618381 Phase I/
Rhabdomyosarcoma 350 FGFR4 inhibitor + CAR-T (ROR1) TKI + CAR-T Orphan + RPDD COG ARST2021 trial
DIPG (Diffuse Intrinsic Pontine Glioma) 300 ONC201 + GD2 CAR-T (CED) + H3K27M p Small molecule RPDD + Breakthr ONC201 expanded acce
Neuroblastoma (High-Risk) 800 Dinutuximab + GD2 CAR-T + Lorlatini Ab + CAR-T + TK Orphan + RPDD ANBL2232 Phase III
Medulloblastoma 500 Sonidegib (SHH) + GD2/B7-H3 CAR-T + SMOi + CAR-T + Orphan + RPDD SJMB21 adaptive tria
Synovial Sarcoma 800 Afamitresgene autoleucel (NY-ESO-1 TCR-T RMAT + Priority BLA submitted 2024
Chordoma 300 GI-6301 (Brachyury vaccine) + Palbo Vaccine + TKI Orphan Drug Phase II NCI
Desmoplastic Small Round Cell Tumor 100 Trabectedin + Temozolomide + anti-I Chemo + TKI Orphan + RPDD NCI MATCH arm
Epithelioid Sarcoma 200 Tazemetostat + Pembrolizumab + Doxo EZH2i + IO Orphan (approve Tazemetostat FDA app
Alveolar Soft Part Sarcoma 100 Atezolizumab (IO) + Cediranib (VEGF IO + TKI Orphan Drug Phase II positive da
Clear Cell Sarcoma 100 Pembrolizumab + Lenvatinib + MET in IO + TKI Orphan Drug NCI trials
PEComa 200 Nab-sirolimus (Fyarro) mTORi nanoparti Full Approval FDA APPROVED 2021
Angiosarcoma 300 Paclitaxel + Pembrolizumab + Bevaci Chemo + IO + an Orphan Drug Phase II trials
Leiomyosarcoma 1500 Trabectedin + Doxorubicin + Olaratu Chemo combo Accelerated App Standard 2nd line

Emerging Screening Technologies

  • Multi-Cancer Early Detection (MCED): cfDNA methylation patterns - Detects: 50+ cancer types (Sensitivity: 51.5% overall, 90%+ for late stage)
  • Circulating Tumor DNA (ctDNA): Tumor mutation detection in blood - Detects: Any with mutations (Sensitivity: 70-90% for advanced)
  • Circulating Tumor Cells (CTCs): Intact tumor cells in blood - Detects: Breast, Prostate, Colorectal (Sensitivity: 30-70%)
  • Exosome/Extracellular Vesicle Analysis: Tumor-derived vesicles with RNA/protein - Detects: Prostate, Lung, Pancreas (research) (Sensitivity: 70-80%)
  • Proteomics/Protein Biomarkers: Multi-protein panels - Detects: Multiple (Sensitivity: Varies by cancer)
  • Breath Analysis (Volatile Organic Compounds): VOC patterns from metabolism - Detects: Lung, Colorectal, others (Sensitivity: 70-85%)
  • AI-Enhanced Imaging: Deep learning on CT/MRI/pathology - Detects: Lung, Breast, Prostate, others (Sensitivity: 90-95%)
  • Methylation Arrays: Genome-wide methylation - Detects: Brain tumors, many others (Sensitivity: 95%+ for classification)

Oral Drug Pipeline (36 Pills for All Cancers)

FDA-Approved Oral Alternatives (12 Available Now)

Cancer Drug Target Dosing Replaces
Ovarian Cancer Olaparib (Lynparza) BRCA1/2 300mg BID oral Platinum maintenance
Ovarian Cancer Niraparib (Zejula) HRD+ 200-300mg QD or Platinum maintenance
Ovarian Cancer Rucaparib (Rubraca) All-comers 600mg BID oral Maintenance after pl
Glioblastoma Vorasidenib (Servier IDH1 R132H 40mg QD oral Watch & wait for low
Liver Cancer (HCC) Lenvatinib (Lenvima) VEGFR/FGFR/RET 8-12mg QD oral First-line HCC
Liver Cancer (HCC) Sorafenib (Nexavar) VEGFR 400mg BID oral First-line HCC
Liver Cancer (HCC) Cabozantinib (Cabome c-MET 60mg QD oral Second-line HCC
Triple-Negative Breast Ca Olaparib (Lynparza) BRCA1/2 300mg BID oral Adjuvant/metastatic
Anaplastic Thyroid Cancer Dabrafenib + Trameti BRAF V600E 150mg BID + 2mg All prior chemo
Anaplastic Thyroid Cancer Selpercatinib (Retev RET fusion 160mg BID oral RET-fusion thyroid
Epithelioid Sarcoma Tazemetostat (Tazver EZH2/INI1 loss 800mg BID oral All prior chemo
PEComa Nab-sirolimus (Fyarr mTOR/TSC IV → oral sirol All prior

Pipeline Oral Drugs (24 in Development)

Cancer Drug Target Phase Est. Approval
Pancreatic Cancer MRTX1133 KRAS G12D Phase I/II 2026-2027
Pancreatic Cancer RMC-9805 (Tri-comple KRAS G12V Phase I 2027-2028
Pancreatic Cancer BI-2865 (pan-KRAS) KRAS-pan Phase I 2027-2028
Glioblastoma Dacomitinib EGFR amplificat Phase II 2026-2027
Small Cell Lung Cancer Talazoparib (Talzenn PARP/DNA damage Phase III (E 2026
Small Cell Lung Cancer Navitoclax + Venetoc BCL-2 Phase I/II 2027
Small Cell Lung Cancer Alisertib Aurora kinase Phase II 2026-2027
Triple-Negative Breast Ca Enzalutamide (Xtandi Androgen recept Phase II 2026
Triple-Negative Breast Ca Ipatasertib AKT pathway Phase III 2025-2026
Pancreatic Ductal Adenoca Sotorasib (Lumakras) KRAS G12C Phase I/II ( 2025-2026
Glioblastoma Erdafitinib (Balvers FGFR3-TACC3 fus Basket trial 2025
Gastric Cancer (HER2-) Futibatinib (Lytgobi FGFR2 Phase II gas 2026
Gastric Cancer (HER2-) Apatinib VEGFR2 FDA filed 2025
Ewing Sarcoma Seclidemstat LSD1 Phase I/II 2026-2027
Synovial Sarcoma Tazemetostat (Tazver EZH2 Phase II sar 2026

Chemo-to-Oral Conversions (24 IV Chemos → Pills)

IV Chemo Oral Alternative Status Efficacy
Cisplatin Satraplatin Phase III (hormone-r Similar to cisplatin
Carboplatin PARP inhibitors (Olaparib FDA APPROVED Superior PFS in BRCA+
Paclitaxel (Taxol) Oraxol (oral paclitaxel + FDA APPROVED 2024 Non-inferior to IV paclit
Docetaxel (Taxotere) ModraDoc006/r (oral docet Phase III Similar to IV docetaxel
Doxorubicin (Adriamy Aldoxorubicin (nanopartic Phase III sarcoma Better tumor penetration
5-Fluorouracil (5-FU Capecitabine (Xeloda) FDA APPROVED Equivalent to IV 5-FU
Gemcitabine LY2334737 (oral gemcitabi Phase II Under investigation
Cytarabine (Ara-C) Oral azacitidine (CC-486) FDA APPROVED Improved OS as maintenanc
Methotrexate IV Oral methotrexate FDA APPROVED Equivalent for low-dose
Vincristine Vinorelbine oral (Navelbi FDA APPROVED Equivalent (NSCLC)
Vinblastine Oral vinorelbine + target Phase II combos Similar activity
Etoposide IV Oral etoposide FDA APPROVED 50% bioavailability (dose

Oral Options for Common Cancers

  • Breast Cancer (HR+): Letrozole, Palbociclib, Fulvestrant → Elacestrant
  • Breast Cancer (HER2+): Tucatinib (Tukysa), Neratinib (Nerlynx), Lapatinib (Tykerb)
  • Colorectal Cancer: Capecitabine, Regorafenib, Trifluridine/tipiracil
  • Prostate Cancer: Enzalutamide, Abiraterone, Olaparib
  • Lung Cancer (NSCLC): Osimertinib, Alectinib, Sotorasib
  • Melanoma: Dabrafenib + Trametinib, Encorafenib + Binimetinib
  • CLL: Ibrutinib, Venetoclax, Acalabrutinib
  • Multiple Myeloma: Lenalidomide, Pomalidomide, Ixazomib

🔬 BEYOND CANCER: All Diseases - IV to Oral Upgrades

63 Total Upgrades | 52 FDA-Approved

This framework discovers oral pill upgrades for ALL major diseases, not just cancer.

Autoimmune Diseases (IV Infusions → Oral Pills)

Disease Current IV/Injectable Oral Upgrade Status
Rheumatoid Arthritis Infliximab (Remicade) IV infus Tofacitinib (Xeljanz FDA APPROVED
Rheumatoid Arthritis Adalimumab (Humira) injection Upadacitinib (Rinvoq FDA APPROVED
Rheumatoid Arthritis Tocilizumab (Actemra) IV Baricitinib (Olumian FDA APPROVED
Psoriasis Ustekinumab (Stelara) injectio Deucravacitinib (Sot FDA APPROVED 20
Psoriatic Arthritis Secukinumab (Cosentyx) injecti Apremilast (Otezla) FDA APPROVED
Ulcerative Colitis Vedolizumab (Entyvio) IV Ozanimod (Zeposia) FDA APPROVED
Ulcerative Colitis Infliximab (Remicade) IV Tofacitinib (Xeljanz FDA APPROVED
Crohn's Disease Adalimumab (Humira) injection Upadacitinib (Rinvoq FDA APPROVED 20

Cardiovascular (Injections → Oral Pills)

Disease Current Injectable Oral Upgrade Status
Atrial Fibrillation / VTE Heparin / Enoxaparin injection Apixaban (Eliquis) FDA APPROVED
VTE Prevention Enoxaparin (Lovenox) injection Rivaroxaban (Xarelto) FDA APPROVED
Heart Failure (HFrEF) IV diuretics + inotropes Sacubitril/Valsartan (Ent FDA APPROVED
Heart Failure Standard therapy Dapagliflozin (Farxiga) FDA APPROVED
Pulmonary Arterial Hypert Epoprostenol (Flolan) IV conti Selexipag (Uptravi) FDA APPROVED
Pulmonary Arterial Hypert Treprostinil SC/IV Treprostinil extended-rel FDA APPROVED

Infectious Diseases (IV Antibiotics/Antivirals → Oral)

Disease Current IV Oral Upgrade Status
HIV Multiple daily pills Biktarvy (BIC/FTC/TAF) FDA APPROVED
HIV Prevention (PrEP) Daily Truvada Lenacapavir (Sunlenca) FDA APPROVED 20
Hepatitis C Interferon + Ribavirin injecti Sofosbuvir/Velpatasvir (E FDA APPROVED
Hepatitis C Peginterferon injections **Glecaprevir/Pibrentasvir ** FDA APPROVED
Hepatitis B Peginterferon alfa injection Tenofovir alafenamide (Ve FDA APPROVED
MRSA Skin Infection Vancomycin IV Linezolid (Zyvox) FDA APPROVED
Osteomyelitis 6 weeks IV antibiotics Oral step-down therapy OVIVA trial pro
C. difficile Infection IV metronidazole Fidaxomicin (Dificid) FDA APPROVED

Neurological Diseases (Injections → Oral)

Disease Current Injectable Oral Upgrade Status
Chronic Migraine Erenumab (Aimovig) injection m Atogepant (Qulipta) FDA APPROVED 20
Episodic Migraine Fremanezumab (Ajovy) injection Rimegepant (Nurtec) FDA APPROVED
Parkinson's Disease Apomorphine SC injection Apomorphine sublingual (K FDA APPROVED 20
Parkinson's OFF Episodes Levodopa/carbidopa intestinal Istradefylline (Nourianz) FDA APPROVED 20
Epilepsy (Status Epilepti IV benzodiazepines Cenobamate (Xcopri) FDA APPROVED 20
ALS Edaravone (Radicava) IV Edaravone oral suspension FDA APPROVED 20

Metabolic & Endocrine (Injections → Oral)

Disease Current Injectable Oral Upgrade Status
Type 2 Diabetes Insulin injections Semaglutide oral (Rybelsu FDA APPROVED 20
Type 2 Diabetes Dulaglutide (Trulicity) inject Tirzepatide oral (in deve Phase III
Obesity Semaglutide (Wegovy) injection **Oral semaglutide (higher ** Phase III for o
Obesity Tirzepatide (Zepbound) injecti Orforglipron Phase III
Osteoporosis Denosumab (Prolia) injection q Alendronate (Fosamax) FDA APPROVED
Severe Osteoporosis Teriparatide (Forteo) daily in Abaloparatide oral (in de Phase II

Hematologic Diseases (IV/Infusions → Oral)

Disease Current IV Oral Upgrade Status
Sickle Cell Disease Blood transfusions Voxelotor (Oxbryta) FDA APPROVED 20
Sickle Cell Disease Hydroxyurea Crizanlizumab oral (in de Phase II
Hemophilia A Factor VIII IV infusions Fitusiran (siRNA) FDA APPROVED 20
Immune Thrombocytopenia Romiplostim (Nplate) SC Eltrombopag (Promacta) FDA APPROVED
Paroxysmal Nocturnal Hemo Eculizumab (Soliris) IV q2wk Danicopan (Voydeya) FDA APPROVED 20
PNH Ravulizumab (Ultomiris) IV Iptacopan (Fabhalta) FDA APPROVED 20

Rare & Genetic Diseases (IV Enzyme Replacement → Oral)

Disease Current IV Oral Upgrade Status
Cystic Fibrosis Inhaled medications + IV antib Elexacaftor/Tezacaftor/Iv FDA APPROVED 20
Fabry Disease Agalsidase beta (Fabrazyme) IV Migalastat (Galafold) FDA APPROVED 20
Gaucher Disease Type 1 Imiglucerase (Cerezyme) IV Eliglustat (Cerdelga) FDA APPROVED 20
Phenylketonuria (PKU) Strict diet + medical foods **Pegvaliase → Sapropterin ** FDA APPROVED
Hereditary Angioedema C1-INH concentrate IV Berotralstat (Orladeyo) FDA APPROVED 20
Transthyretin Amyloidosis Patisiran (Onpattro) IV q3wk Tafamidis (Vyndaqel) FDA APPROVED 20

Psychiatric Disorders

Disease Current Treatment Oral Upgrade Status
Treatment-Resistant Depre Esketamine (Spravato) nasal Psilocybin (in developmen Phase III (Brea
Treatment-Resistant Depre IV ketamine infusions Oral ketamine compounds Phase II
Schizophrenia Paliperidone LAI monthly Lumateperone (Caplyta) FDA APPROVED 20
ADHD Standard stimulants Viloxazine ER (Qelbree) FDA APPROVED 20

Framework Tools (62 Total)

By Category

Category Tools Purpose
Literature PubMed search, citation analysis Evidence gathering
Clinical Trials Trial search, eligibility matching Patient enrollment
Genomics Variant analysis, pathway mapping Precision medicine
Drug Discovery Target identification, compound screening New drug development
Biomarkers Biomarker panels, predictive markers Patient stratification
Treatment Response prediction, toxicity analysis Treatment optimization
Curative Biotech CAR-T, mRNA, CRISPR, oncolytic virus Next-gen therapies
CAD Target discovery, FDA proposal generation Accelerated approval
Oral Therapy Pill alternatives to chemo Patient convenience
Gap Analysis Unmet needs, emerging solutions R&D prioritization

Quick Commands

# Match patient to curative therapy
python cicd/patient_match.py --cancer "DLBCL" --biomarkers "CD19+"

# Find oral alternative to chemo
python cicd/patient_match.py --cancer "NSCLC" --biomarkers "EGFR T790M"

# Run full analysis
python cicd/runner.py

Installation

git clone https://github.com/ClandestineAI/cancer-core-agentic-framework.git
cd cancer-core-agentic-framework
npm install
npm run build

API Keys (Optional)

export TAVILY_API_KEY="your-key"  # For real-time research

Local CI/CD

This framework includes local CI/CD that auto-runs on every commit:

  • Build: TypeScript compilation and type checking
  • Validate: Verify all therapeutic data (CAR-T, mRNA, CRISPR, oral therapies)
  • Test: Run test suite
  • README: Auto-regenerate this documentation

License

MIT - For research and clinical decision support. Not a substitute for professional medical advice.


This README auto-generated from framework data. See cicd/generate_readme.py

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⬡ Oncology CADD · OSINT Interactive drug-discovery triage on public data

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